Basic Peptide Information

DICL ID
DICL_Pep_01109
Ion Channel
Neuronal acetylcholine receptor subunit alpha-9/alpha-10
Peptide Function
Antagonist
Gene Name
CHRNA9/CHRNA10

Activity Data (nM)

IC50
1.5 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
GCCSDPRCRYRCR
Peptide UniProt Accession
UniParc
UPI0000D8554A
Peptide Synonyms/Alias
Not available
Peptide Species
Conus regius (Crown cone)
Peptide Name
Alpha-conotoxin RgIA
CAS Number
Not available

Experimental Conditions

pH
pH 7.1 to 7.5
Holding Potential (mV)
Not mention
Temperature
Not mention
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available